X-Rx has a robust drug pipeline with multiple programs in development.

The X-Rx pipeline features:

  • ATX, an orally bioavailable small molecule inhibitor of autotaxin, currently in IND enabling studies.
  • BTKwt, a highly selective, orally bioavailable irreversible antagonist of Bruton’s Tyrosine Kinase (BTK). The program was partnered with a top-tier biotech in China in 2015.
  • Multiple leads at discovery phase in the following target areas: protein-protein interactions, kinases and GPCRs
  • Access to new screens for novel targets